CS-2100

CAT: 0804-HY-108493-01Size: 5 mgDry Ice: NoHazardous: No
CAT#:0804-HY-108493-01Size:5 mg
Selected
PRICE
AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Product image 1
1 / 1
Description
CS-2100 (Compound 10b) is a potent, selective, orally active and S1P3-sparing S1P1 agonist with an EC50 of 4.0 nM for human S1P1. CS-2100 shows in vivo immunosuppressive efficacy in rats with an ID50 (infective dose) of 0.407 mg/kg for HvGR[1].
CAS Number
[913827-99-3]
UNSPSC
12352005
Hazard Statement
H302-H315-H319
Target
LPL Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
COVID-19-immunoregulation
Field of Research
Inflammation/Immunology
Assay Protocol
https://www.medchemexpress.com/cs-2100.html
Purity
99.12
Solubility
DMSO : 12.5 mg/mL (ultrasonic; warming; heat to 60°C)
Smiles
O=C(C1CN(CC2=CC(CC)=C(C3=NOC(C4=CC=C(OC5=CC=CC=C5)C=C4)=N3)S2)C1)O
Molecular Formula
C25H23N3O4S
Molecular Weight
461.53
Precautions
P264-P270-P280-P302+P352-P305+P351+P338-P330-P362+P364-P501
References & Citations
[1]Nakamura T, et al. Discovery of CS-2100, a potent, orally active and S1P3-sparing S1P1 agonist. Bioorg Med Chem Lett. 2012 Feb 15;22 (4) :1788-92.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported

Related Products

CatalogName
HY-101824NC-2100
HY-120219-01TU-2100
HY-14976CS-0777
HY-100413CS-526
HY-107163CS 461
HY-175198Cs-2d
HY-19633ACS-003
HY-P6306-01CS-6253
HY-106888ACS-722
HY-P6306A-01CS-6253 (TFA)

Alternative Products

CatalogName
MF-0050396-01CS 2100
MF-0050258-01TU-2100
MF-0038280W-2100
MBS5812734NC-2100
4002100WSC-2100 MyMiniAspirator
EGF2100-1000EnoGeneFec™ 2100 Transfection Reagent
E36G2100DNAfectin™ 2100 Transfection Reagent
AUT4502Prestige Autoclave 2100 Extended
MBS8579500-01EnoGeneFec 2100 Transfection Reagent
MBS8580096-01DNAfectin 2100 Transfection Reagent

Popular Products