Products for Research Use Only
RegisterLogin

CB2R antagonist 3

CAT: 0804-HY-152581-01Size: 5 mgDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0804-HY-152581-01Size:5 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
Description
CB2R antagonist 3 is a selective antagonist of cannabinoid type 2 receptor (CB2R). CB2R antagonist 3 has high affinity for human CB2R and specific selectivity for CB1R. CB2R antagonist 3 can be combined with CB65 , the activator of CB2R. CB2R antagonist 3 effectively up-regulates the expression of anti-inflammatory cytokines and down-regulates the expression of pro-inflammatory cytokines[1].
UNSPSC
12352005
Target
Cannabinoid Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
COVID-19-immunoregulation
Field of Research
Inflammation/Immunology
Assay Protocol
https://www.medchemexpress.com/cb2r-antagonist-3.html
Purity
98.08
Solubility
DMSO : 100 mg/mL (ultrasonic; warming; heat to 60°C)
Smiles
CCCCCNC1=C(C=C(C=C1)CCCCC)C(NC23CC4CC(C3)CC(C2)C4)=O
Molecular Formula
C27H42N2O
Molecular Weight
410.64
References & Citations
[1]Graziano G, et al. N-adamantyl-anthranil amide derivatives: New selective ligands for the cannabinoid receptor subtype 2 (CB2R) . Eur J Med Chem. 2023 Feb 15;248:115109.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
CB2

Related Products

CatalogName
HY-175784CB2R antagonist 4
HY-149644CB2R agonist 3
HY-152254-01CB2R/FAAH modulator-3
HY-100328CB2R-IN-1
HY-131004-01CB2R PAM
HY-155481CB2 receptor antagonist 3
HY-152576CB2R agonist 1
HY-175730CB2R ligand-1
HY-155336CB2R agonist 2
HY-147532CB2R probe 1

Alternative Products

CatalogName
GTR19273374-01CB2R antagonist 4
T73326-01CB2R-IN-3
MBS5798058CB2R PAM
T10697-01CB2R-IN-1
T82770-01CB2R agonist 2
T82769-01CB2R agonist 3
A12306-50CB2R-IN-1 50mg
A12306-5CB2R-IN-1 5mg
MBS5815111CB2R agonist 1
GTR19264341-01CB2R agonist 4

Popular Products