CB2R agonist 4

CAT: 0804-HY-175481Size: 1 EachDry Ice: NoHazardous: No
CAT#:0804-HY-175481Size:1 Each
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Description
CB2R agonist 4 is a cannabinoid receptor 2 (CB2R) agonist with an EC50 value of 6.9 μM. CB2R agonist 4 can induce cell apoptosis, ROS production and protein misfolding. CB2R agonist 4 shows cytotoxicity to a panel of tumor cell lines. CB2R agonist 4 can be used for the research of cancer[1].
CAS Number
[182496-82-8]
UNSPSC
12352005
Target
Apoptosis; Cannabinoid Receptor; Reactive Oxygen Species (ROS)
Related Pathways
Apoptosis; GPCR/G Protein; Immunology/Inflammation; Metabolic Enzyme/Protease; Neuronal Signaling; NF-κB
Applications
Cancer-programmed cell death
Field of Research
Cancer
Smiles
O=C(OCC1=CC=CC=C1)[C@@H](N2C(C3=CC=CC=C3NC2=O)=O)CC(C)C
Molecular Formula
C21H22N2O4
Molecular Weight
366.41
References & Citations
[1]Ciaglia T, et al. Untargeted Diversity-Oriented Synthesis for the Discovery of New Antitumor Agents: An Integrated Approach of Inverse Virtual Screening, Bioinformatics, and Omics for Target Deconvolution. J Med Chem. 2025 Aug 14;68 (15) :16483-16517.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
CB2

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