Products for Research Use Only
RegisterLogin

A3AR antagonist 3

CAT: 0804-HY-120652-01Size: 500 µgDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0804-HY-120652-01Size:500 µg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
Description
A3AR antagonist 3 (compound 21) is a selective A3 adenosine receptor (A3AR) antagonist with a Ki of 37 nM. A3AR antagonist 3 shows >60-fold selectivity in comparison to A1 and A2A adenosine receptors[1].
CAS Number
863202-33-9
UNSPSC
12352005
Hazard Statement
H302-H315-H319-H335
Target
Adenosine Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
COVID-19-immunoregulation
Field of Research
Inflammation/Immunology
Assay Protocol
https://www.medchemexpress.com/a3ar-antagonist-3.html
Solubility
10 mM in DMSO
Smiles
[H][C@@]12[C@H]([C@@](C2)([H])CC1)NC3=C4N=CNC4=NC(NC5=CC=CC=C5)=N3
Molecular Formula
C17H18N6
Molecular Weight
306.37
Precautions
P261-P264-P270-P271-P280-P302+P352-P304+P340-P305+P351+P338-P330-P362+P364-P403+P233-P405-P501
References & Citations
[1]Melissa Perreira, et al. "Reversine" and its 2-substituted adenine derivatives as potent and selective A3 adenosine receptor antagonists. J Med Chem. 2005 Jul 28;48 (15) :4910-8.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
Adenosine A1 receptor (A1R) ; Adenosine A2A receptor (A2AR) ; Adenosine A3 receptor (A3R)

Related Products

CatalogName
HY-179671A3AR antagonist 6
HY-134555-01A3AR antagonist 4
HY-164621-01A3AR antagonist 5
HY-12099A3AR antagonist 2
HY-146457A3AR antagonist 1
HY-158179A3AR agonist 3
HY-151899A3AR modulator 1
HY-158180A3AR agonist 4
HY-155184A3AR agonist 2
HY-155183A3AR agonist 1

Alternative Products

CatalogName
MBS5806624A3AR antagonist 1
MBS5814926A3AR antagonist 2
GTR19238885-01A3AR antagonist 5
GTR19274086-01A3AR antagonist 6
T85531-01A3AR agonist 3
MBS5816916A3AR modulator 1
GTR19235731-01A3AR agonist 4
MBS5821035A3AR agonist 2
MBS5821034A3AR agonist 1
GTR19235730-01A3AR agonist 5

Popular Products