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Masupirdine free base

CAT: 0931-T11948-01Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0931-T11948-01Size:1 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
701205-60-9
Target
5-HT Receptor
Related Pathways
GPCR/G Protein, Neuroscience
Purity
0.9965
Bioactivity
Masupirdine free base (SUVN-502 free base) is an orally available 5-HT6 receptor antagonist that crosses the blood-brain barrier, with a Ki value of 2.04 nM for the human 5-HT6 receptor. It is potent and selective, inhibiting multiple targets, and can be used in the study of neurological disorders such as Alzheimer's disease.
Smiles
O=S(=O)(C=1C=CC=CC1Br)N2C=C(C=3C=C(OC)C=CC32)CN4CCN(C)CC4
Molecular Formula
C21H24BrN3O3S
Molecular Weight
478.4
Shipping Conditions
Ice Packs
Storage Temperature
-20°C