Products for Research Use Only

EST64454 free base

CAT: 0931-T70908-01Size: 25 mgDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0931-T70908-01Size:25 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
CAS Number
1351438-26-0
Target
Others, Sigma receptor
Related Pathways
GPCR/G Protein, Others
Bioactivity
EST64454 is a σ1 receptor (σ1R) antagonist clinical candidate for the treatment of pain. EST64454 shows an outstanding aqueous solubility, which together with its high permeability in Caco-2 cells will allow its classification as a BCS class I compound. It also shows high metabolic stability.
Smiles
C(OCCN1CCN(C(C)=O)CC1)C2=NN(C=C2)C3=CC(F)=C(F)C=C3
Molecular Formula
C18H22F2N4O2
Molecular Weight
364.39
Shipping Conditions
Ice Packs
Storage Temperature
-20°C