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AR-M 1000390

CAT: 0804-HY-101039Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-101039Size:1 Each
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
AR-M 1000390 is an exceptionally selective, potent δ opioid receptor agonist with an EC50 of 7.2±0.9 nM for δ agonist potency.
CAS Number
209808-01-5
UNSPSC
12352005
Target
Opioid Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/ar-m-1000390.html
Solubility
10 mM in DMSO
Smiles
O=C(N(CC)CC)C1=CC=C(/C(C2=CC=CC=C2)=C3CCNCC/3)C=C1
Molecular Formula
C23H28N2O
Molecular Weight
348.48
References & Citations
[1]Wei ZY, et al. N, N-Diethyl-4- (phenylpiperidin-4-ylidenemethyl) benzamide: a novel, exceptionally selective, potent delta opioid receptor agonist with oral bioavailability and its analogues. J Med Chem. 2000 Oct 19;43 (21) :3895-905.|[2]Otieno MA, et al. Mechanistic investigation of N, N-diethyl-4- (phenyl-piperidin-4-ylidenemethyl) -benzamide-inducedinsulin depletion in the rat and RINm5F cells. Toxicol Sci. 2008 Sep;105 (1) :221-9.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported

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Alternative Products

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T89183-01AR-M 1000390
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A21911-25AR-M 1000390 hydrochloride 25mg
A21911-10AR-M 1000390 hydrochloride 10mg
A21911-5AR-M 1000390 hydrochloride 5mg
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