SRC-3-IN-2
CAT:
804-HY-163469
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- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No


SRC-3-IN-2
UNSPSC Description:
SRC-3-IN-2 (SI-12 6c)is an orally active steroid receptor coactivator 3 (SRC-3) inhibitor. SRC-3-IN-2 has antitumor activity[1].Target Antigen:
SrcType:
Reference compoundRelated Pathways:
Protein Tyrosine Kinase/RTKApplications:
Cancer-programmed cell deathField of Research:
CancerAssay Protocol:
https://www.medchemexpress.com/src-3-in-2.htmlSolubility:
10 mM in DMSOSmiles:
C/C(C1=NC=C(C=C1)F)=N\N=C2N(C3=C(N\2)C=C(F)C(F)=C3)CMolecular Weight:
319.28References & Citations:
[1] Lu D, et al. Lead Compound Development of SRC-3 Inhibitors with Improved Pharmacokinetic Properties and Anticancer Efficacy. J Med Chem. 2024 Mar 29.Shipping Conditions:
Room temperatureClinical Information:
No Development Reported