SRC-3-IN-2

• Description:

  SRC-3-IN-2 (SI-12 6c) is an orally active steroid receptor coactivator 3 (SRC-3) inhibitor. SRC-3-IN-2 has antitumor activity[1].

• UNSPSC:

  12352005

• Target:

  Src

• Type:

  Reference compound

• Related Pathways:

  Protein Tyrosine Kinase/RTK

• Applications:

  Cancer-programmed cell death

• Field of Research:

  Cancer

• Assay Protocol:

  https://www.medchemexpress.com/src-3-in-2.html

• Concentration:

  10mM

• Purity:

  96.32

• Solubility:

  DMSO : 25 mg/mL (ultrasonic)

• Smiles:

  CN1C2=CC(F)=C(F)C=C2N/C1=N\N=C(C3=CC=C(C=N3)F)/C

• Molecular Formula:

  C15H12F3N5

• Molecular Weight:

  319.28

• References & Citations:

  [1] Lu D, et al. Lead Compound Development of SRC-3 Inhibitors with Improved Pharmacokinetic Properties and Anticancer Efficacy. J Med Chem. 2024 Mar 29.

• Shipping Conditions:

  Room Temperature

• Storage Conditions:

  4°C (Powder, protect from light)

• Scientific Category:

  Reference compound1

• Clinical Information:

  No Development Reported

• CAS Number:

  [3074959-44-4]