CGP-53153

CAT: 0804-HY-U00125Size: 1 EachDry Ice: NoHazardous: No

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CAT#:0804-HY-U00125Size:1 Each

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Description

CGP-53153 is a steroidal inhibitor of 5 alpha reductase with IC50s of 36 and 262 nM in rat and human prostatic tissue, respectively.

CAS Number

149281-19-6

UNSPSC

12352005

Target

5 alpha Reductase

Type

Reference compound

Related Pathways

Metabolic Enzyme/Protease

Applications

Metabolism-sugar/lipid metabolism

Field of Research

Endocrinology

Assay Protocol

https://www.medchemexpress.com/CGP-53153.html

Solubility

10 mM in DMSO

Smiles

C[C@@]1([C@H]2C(NC(C)(C)C#N)=O)[C@](CC2)([H])[C@@](CC[C@](N3)([H])[C@@]4(C=CC3=O)C)([H])[C@]4([H])CC1

Molecular Formula

C23H33N3O2

Molecular Weight

383.53

References & Citations

[1]H?usler A, et al. CGP-53153: a new potent inhibitor of 5alpha-reductase. J Steroid Biochem Mol Biol. 1996 Feb;57 (3-4) :187-95.

Shipping Conditions

Room temperature

Scientific Category

Reference compound1

Clinical Information

No Development Reported

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