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GR 89696

CAT: 0804-HY-107747-01Size: 5 mgDry Ice: NoHazardous: No
CAT#:0804-HY-107747-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
GR 89696 is a highly selective κ2 opioid receptor agonist with potential to prevent pruritus[1].
CAS Number
[126766-32-3]
UNSPSC
12352005
Target
Opioid Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
COVID-19-immunoregulation
Field of Research
Inflammation/Immunology
Assay Protocol
https://www.medchemexpress.com/gr-89696.html
Concentration
10mM
Purity
99.88
Solubility
DMSO : ≥ 50 mg/mL
Smiles
OC(/C=C/C(O)=O)=O.ClC(C=C1CC(N2C(CN(CC2)C(OC)=O)CN3CCCC3)=O)=C(C=C1)Cl
Molecular Formula
C23H29Cl2N3O7
Molecular Weight
530.40
References & Citations
[1]Mei-Chuan Ko, et al. Effects of atypical kappa-opioid receptor agonists on intrathecal morphine-induced itch and analgesia in primates. J Pharmacol Exp Ther. 2009 Jan;328 (1) :193-200. |[2]A Barber, et al. Effects of GR-89696 and the novel peripherally selective OP2 agonists, EMD-61569 and EMD-61747, against focal cerebral ischemia in the rat. Methods Find Exp Clin Pharmacol. 1999 Mar;21 (2) :105-13
Shipping Conditions
Room Temperature
Storage Conditions
4°C (Powder, sealed storage, away from moisture)
Scientific Category
Reference compound1
Clinical Information
No Development Reported

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