THR-β modulator-1
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No


THR-β modulator-1
Description:
THR-β modulator-1 (compound 1a) is a potent thyroid hormone receptor β modulator. THR-β modulator-1 can be used in research of thyroid hormone receptor related disorders[1].UNSPSC:
12352005Target:
Thyroid Hormone ReceptorType:
Reference compoundRelated Pathways:
Vitamin D Related/Nuclear ReceptorApplications:
Metabolism-protein/nucleotide metabolismField of Research:
EndocrinologyAssay Protocol:
https://www.medchemexpress.com/thr-β-modulator-1.htmlSolubility:
10 mM in DMSOSmiles:
O=C1C2=C(CC[C@H]2C)C(OC3=C(Cl)C=C(N4N=C(N)C(NC4=O)=O)C=C3Cl)=NN1Molecular Formula:
C17H14Cl2N6O4Molecular Weight:
437.24References & Citations:
[1]David CM, et, al. Bicyclic pyridazinones and methods of use thereof. WO2022099060A2.Shipping Conditions:
Room temperatureScientific Category:
Reference compound1Clinical Information:
No Development ReportedCAS Number:
2770373-00-5
