PPARγ agonist 1

PPARγ agonist 1

• CAS Number: 3032632-09-7
• UNSPSC Description: PPARγ agonist 1 (compound 15) is a potent agonist of PPARγ. PPARγ agonist 1 shows high efficacy to activate hPPARγ without raising a full agonism and probably avoiding adverse effects. PPARγ agonist 1 has the potential for the research of cardiovascular diseases associated with metabolic disorders[1].
• Target Antigen: PPAR
• Type: Reference compound
• Related Pathways: Cell Cycle/DNA Damage;Metabolic Enzyme/Protease;Vitamin D Related/Nuclear Receptor
• Applications: Metabolism-protein/nucleotide metabolism
• Field of Research: Metabolic Disease; Cardiovascular Disease
• Assay Protocol: https://www.medchemexpress.com/pparγ-agonist-1.html
• Solubility: 10 mM in DMSO
• Smiles: C/C(CC/C=C(C(NC1=CC=CC=C1)=O)\C)=C\CCC2(CCC3=C(O2)C=CC(OCC4=CC=CC=C4)=C3)C
• Molecular Weight: 509.68
• References & Citations: [1]Vila L, et al. Synthesis and biological studies of "Polycerasoidol" and "trans-δ-Tocotrienolic acid" derivatives as PPARα and/or PPARγ agonists. Bioorg Med Chem. 2022;53:116532.
• Shipping Conditions: Room temperature
• Clinical Information: No Development Reported