5-HT6/5-HT2A receptor ligand-1

5-HT6/5-HT2A receptor ligand-1

• CAS Number: 2411088-07-6
• UNSPSC Description: 5-HT6/5-HT2A receptor ligand-1 (compound 33) is a dual 5-HT6/5-HT2A receptor antagonist, with a Ki of 2 nM and 11 nM, respectively. 5-HT6/5-HT2A receptor ligand-1 has the potential for neurological and psychiatric disorders research[1].
• Target Antigen: 5-HT Receptor
• Type: Reference compound
• Related Pathways: GPCR/G Protein;Neuronal Signaling
• Applications: Neuroscience-Neuromodulation
• Field of Research: Neurological Disease
• Assay Protocol: https://www.medchemexpress.com/5-ht6-5-ht2a-receptor-ligand-1.html
• Solubility: 10 mM in DMSO
• Smiles: OC1=CC=C(C2=CC=C(CNCCC3=CNC4=C3C=C(F)C=C4)O2)C=C1
• Molecular Weight: 350.39
• References & Citations: [1]Staroń J, et, al. Virtual screening-driven discovery of dual 5-HT 6/5-HT 2A receptor ligands with pro-cognitive properties. Eur J Med Chem. 2020 Jan 1;185:111857.
• Shipping Conditions: Room temperature
• Clinical Information: No Development Reported