5-HT2A receptor agonist-3
CAT:
804-HY-153912-01
Size:
1 mg
Price:
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- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No
5-HT2A receptor agonist-3
- CAS Number: 1391499-52-7
- UNSPSC Description: 5-HT2A receptor agonist-3 is the most selective agonist for the human 5-HT2A receptor yet discovered, with a Ki of 2.5 nM, and with 124-fold selectivity for 5-HT2A over the structurally similar 5-HT2C receptor[1].
- Target Antigen: 5-HT Receptor
- Type: Reference compound
- Related Pathways: GPCR/G Protein;Neuronal Signaling
- Applications: Neuroscience-Neuromodulation
- Field of Research: Others
- Assay Protocol: https://www.medchemexpress.com/5-ht2a-receptor-agonist-3.html
- Solubility: 10 mM in DMSO
- Smiles: COC1=C([C@H]2N[C@@H](CCC2)CC3=C(C=C(C(OC)=C3)Br)OC)C=CC=C1
- Molecular Weight: 420.34
- References & Citations: [1]Juncosa JI Jr, et al. Extensive rigid analogue design maps the binding conformation of potent N-benzylphenethylamine 5-HT2A serotonin receptor agonist ligands. ACS Chem Neurosci. 2013;4(1):96-109.
- Shipping Conditions: Room Temperature
- Clinical Information: No Development Reported