PF-184298
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No


PF-184298
UNSPSC Description:
PF-184298 is a dual serotonin/noradrenaline reuptake inhibitor with IC50 of 6 nM and 21 nM, respectively[1].Target Antigen:
OthersType:
Reference compoundRelated Pathways:
OthersApplications:
Neuroscience-NeuromodulationField of Research:
Cardiovascular DiseaseAssay Protocol:
https://www.medchemexpress.com/pf-184298.htmlSolubility:
10 mM in DMSOSmiles:
O=C(C1=CC=CC(Cl)=C1Cl)N([C@@H]2CNCC2)CC(C)CMolecular Weight:
315.24References & Citations:
[1]Anthony Harrison , et al. Case studies addressing human pharmacokinetic uncertainty using a combination of pharmacokinetic simulation and alternative first in human paradigms. Clinical Trial Xenobiotica. 2012 Jan;42(1):57-74.Shipping Conditions:
Room temperatureClinical Information:
No Development ReportedCAS Number:
813447-40-4
