AT-127
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No


AT-127
UNSPSC Description:
AT-127 is a NOP receptor partial agonist, stimulating NOP/G-protein interaction in a concentration dependent manner[1].Target Antigen:
Opioid ReceptorType:
Reference compoundRelated Pathways:
GPCR/G Protein;Neuronal SignalingApplications:
Neuroscience-NeuromodulationField of Research:
Neurological DiseaseAssay Protocol:
https://www.medchemexpress.com/at-127.htmlSolubility:
10 mM in DMSOSmiles:
O=C1N(C2CCN([C@H]3CC[C@H](CC3)C(C)C)CC2)C4=CC=CC=C4/C1=N/OMolecular Weight:
369.50References & Citations:
[1]Federica Ferrari, et al. In vitro functional characterization of novel nociceptin/orphanin FQ receptor agonists in recombinant and native preparations. Eur J Pharmacol. 2016 Dec 15:793:1-13.Shipping Conditions:
Room temperatureClinical Information:
No Development ReportedCAS Number:
2099680-72-3
