PK44 (phosphate)

• UNSPSC Description:

  PK44 phosphate is a potent dipeptidyl peptidase IV (DPP-IV) inhibitor with an IC50 value of 15.8 nM[1].

• Target Antigen:

  Dipeptidyl Peptidase

• Type:

  Reference compound

• Related Pathways:

  Metabolic Enzyme/Protease

• Applications:

  Metabolism-protein/nucleotide metabolism

• Field of Research:

  Metabolic Disease

• Assay Protocol:

  https://www.medchemexpress.com/pk44-phosphate.html

• Solubility:

  10 mM in DMSO

• Smiles:

  O=P(O)(O)O.FC(F)(C1=NN=C2N1CCN(C(C[C@H](N)CC(C3=CC=C4F)=NNC3=C4F)=O)C2)F

• Molecular Weight:

  527.34

• References & Citations:

  [1]Adrian Maddaford, et al. Indazoles for use as dpp-iv inhibitors. WO2008040995A1 (compound 67)

• Shipping Conditions:

  Room temperature

• Clinical Information:

  No Development Reported

• CAS Number:

  1017682-66-4