PK44 (phosphate)

• Description :

  PK44 phosphate is a potent dipeptidyl peptidase IV (DPP-IV) inhibitor with an IC50 value of 15.8 nM[1].

• UNSPSC :

  12352005

• Target :

  Dipeptidyl Peptidase

• Type :

  Reference compound

• Related Pathways :

  Metabolic Enzyme/Protease

• Applications :

  Metabolism-protein/nucleotide metabolism

• Field of Research :

  Metabolic Disease

• Assay Protocol :

  https://www.medchemexpress.com/pk44-phosphate.html

• Solubility :

  10 mM in DMSO

• Smiles :

  O=P(O)(O)O.FC(F)(C1=NN=C2N1CCN(C(C[C@H](N)CC(C3=CC=C4F)=NNC3=C4F)=O)C2)F

• Molecular Formula :

  C17H19F5N7O5P

• Molecular Weight :

  527.34

• References & Citations :

  [1]Adrian Maddaford, et al. Indazoles for use as dpp-iv inhibitors. WO2008040995A1 (compound 67)

• Shipping Conditions :

  Room temperature

• Scientific Category :

  Reference compound1

• Clinical Information :

  No Development Reported

• Isoform :

  DPP-4

• CAS Number :

  [1017682-66-4]