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CGP 39551

CAT: 0804-HY-107703Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-107703Size:1 Each
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Description
CGP 39551 is a potent, orally active, competitive N-methyl-D-aspartate (NMDA) receptor antagonist with potent anticonvulsant activity[1]. CGP 39551 shows measurable inhibitory activity at both L-[3H]-glutamate (Ki=8.4 μM) [2].
CAS Number
127910-32-1
UNSPSC
12352211
Hazard Statement
H301
Target
IGluR
Type
Reference compound
Related Pathways
Membrane Transporter/Ion Channel; Neuronal Signaling
Applications
Neuroscience-Neurodegeneration
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/cgp-39551.html
Solubility
10 mM in DMSO
Smiles
CCOC(C(N)/C=C(C)/CP(O)(O)=O)=O
Molecular Formula
C8H16NO5P
Molecular Weight
237.19
Precautions
P264-P270-P330-P405-P501
References & Citations
[1]G E Fagg, et al. CGP 37849 and CGP 39551: novel competitive N-methyl-D-aspartate receptor antagonists with potent oral anticonvulsant activity. Prog Clin Biol Res. 1990;361:421-7.|[2]G E Fagg, et al. CGP 37849 and CGP 39551: novel and potent competitive N-methyl-D-aspartate receptor antagonists with oral activity. Br J Pharmacol. 1990 Apr;99 (4) :791-7.|[3]R Dall'Olio, et al. Chronic neonatal blockade of N-methyl-D-aspartate receptor by CGP 39551 increases dopaminergic function in adult rat. Neuroscience. 1994 Nov;63 (2) :451-5.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
NMDA Receptor

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