Products for Research Use Only
RegisterLogin

GT-2016

CAT: 0804-HY-107559Size: 1 EachDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0804-HY-107559Size:1 Each
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
Description
GT-2016 is a potent, selective, and brain penetrant histamine H3 receptor antagonist with a Ki of 43.8 nM. GT-2016 displays selectivity against H1 and H2 receptors, and has non-active against histamine methyltransferase[1].
CAS Number
152241-24-2
UNSPSC
12352005
Target
Histamine Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Immunology/Inflammation; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/gt-2016.html
Solubility
10 mM in DMSO
Smiles
O=C(N1CCC(C2=CNC=N2)CC1)CCCCC3CCCCC3
Molecular Formula
C19H31N3O
Molecular Weight
317.47
References & Citations
[1]C E Tedford, et al. Pharmacological characterization of GT-2016, a non-thiourea-containing histamine H3 receptor antagonist: in vitro and in vivo studies. J Pharmacol Exp Ther. 1995 Nov;275 (2) :598-604.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
H3 Receptor

Related Products

CatalogName
HY-154944-01JG-2016
HY-157479DPI-2016
HY-139699GT-055
HY-114381-01GT 949
HY-139698GT-1
HY-158432-01GT-653
HY-174311-01GT-02216
HY-10016-01E 2012
HY-150644-01S07-2010
HY-W725179-01VK-2019

Alternative Products

CatalogName
B7049-5GT 2016
573568GT-2016
T86299-01DPI-2016
T82008-01JG-2016
C0178γ-GT (GAMMA GT)

Popular Products