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CGP 56999

CAT: 0804-HY-123222Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-123222Size:1 Each
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
CGP 56999 is a potent antagonist GABA (B) receptor, with the IC50 of 0.002 μM. CGP 56999 increased the levels of BDNF mRNA in the brain in vivo and in vitro[1].
CAS Number
153994-97-9
UNSPSC
12352005
Target
GABA Receptor
Type
Reference compound
Related Pathways
Membrane Transporter/Ion Channel; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/cgp-56999.html
Smiles
O=C(O)C1=CC=CC([C@H](NC[C@H](O)CP(O)(CC2CCCCC2)=O)C)=C1
Molecular Formula
C19H30NO5P
Molecular Weight
383.42
References & Citations
[1]H. Bittiger, et al. GABAB Receptor Antagonists: Potential Therapeutic Applications. In: Tanaka, C., Bowery, N.G. (eds) GABA: Receptors, Transporters and Metabolism. Advances in Pharmacological Sciences. Birkhäuser Basel.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported