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Mardepodect (succinate)

CAT: 0804-HY-10030Size: 1 EachDry Ice: NoHazardous: No
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CAT#:0804-HY-10030Size:1 Each
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Description
Mardepodect succinate (PF-2545920 succinate) is a potent and specific phosphodiesterase 10A (PDE10A) inhibitor with potential activity in the treatment of schizophrenia. Mardepodect succinate has been further optimized to improve brain penetration and compound-like properties for use in schizophrenia research[1].
CAS Number
1037309-45-7
Product Name Alternative
PF-2545920 (succinate)
UNSPSC
12352005
Target
Phosphodiesterase (PDE)
Type
Reference compound
Related Pathways
Metabolic Enzyme/Protease
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/mardepodect-succinate.html
Smiles
CN(N=C1C2=CC=C(OCC3=NC4=CC=CC=C4C=C3)C=C2)C=C1C5=CC=NC=C5.O=C(O)CCC(O)=O
Molecular Formula
C29H26N4O5
Molecular Weight
510.54
References & Citations
[1]Discovery of a novel class of phosphodiesterase 10A inhibitors and identification of clinical candidate 2-[4- (1-methyl-4-pyridin-4-yl-1H-pyrazol-3-yl) -phenoxymethyl]-quinoline (PF-2545920) for the treatment of schizophrenia
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
Phase 2