Succinate/succinate receptor antagonist 1

CAT:
804-HY-150205-01
Size:
5 mg
  • Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
  • Dry Ice Shipment: No
Succinate/succinate receptor antagonist 1 - image 1

Succinate/succinate receptor antagonist 1

  • UNSPSC Description:

    Succinate/succinate receptor antagonist 1 (compound 7a) is a succinate/succinate receptor antagonist. Succinate/succinate receptor antagonist 1 blocks succinate signaling in gingival tissue. Succinate/succinate receptor antagonist 1 inhibits the activation of succinate receptor 1 (SucnRl) with an IC50 value of 20 μΜ. Succinate/succinate receptor antagonist 1 can be used for the research of periodontal disease[1].
  • Target Antigen:

    Others
  • Type:

    Reference compound
  • Related Pathways:

    Others
  • Applications:

    COVID-19-immunoregulation
  • Field of Research:

    Inflammation/Immunology
  • Assay Protocol:

    https://www.medchemexpress.com/succinate-succinate-receptor-antagonist-1.html
  • Solubility:

    DMSO : 25 mg/mL (ultrasonic)
  • Smiles:

    O=C(NC)CC1=CC=C(C2=NC3=NC=CC=C3C=C2)C=C1
  • Molecular Weight:

    277.32
  • References & Citations:

    [1]LI, Xin, et al. PERIODONTAL DISEASE THERAPY. WO2019136022. 2020.
  • Shipping Conditions:

    Room Temperature
  • Clinical Information:

    No Development Reported
  • CAS Number:

    2361972-29-2