MSX-122

• UNSPSC Description:

  MSX-122 is an orally active partial antagonist of CXCR4, inhibiting CXCR4/CXCL12 actions, with an IC50 of ～10 nM. MSX-122 has anti-inflammatory and anti-metastatic activity.

• Target Antigen:

  CXCR

• Type:

  Reference compound

• Related Pathways:

  GPCR/G Protein;Immunology/Inflammation

• Field of Research:

  Cancer; Inflammation/Immunology; Endocrinology

• Assay Protocol:

  https://www.medchemexpress.com/MSX-122.html

• Smiles:

  C1(CNC2=NC=CC=N2)=CC=C(CNC3=NC=CC=N3)C=C1

• Molecular Weight:

  292.34

• References & Citations:

  [1]Liang Z, et al. Development of a unique small molecule modulator of CXCR4. PLoS One. 2012;7(4):e34038.

• Shipping Conditions:

  Room Temperature

• CAS Number:

  897657-95-3