PSB-1115

• Description:

  PSB-1115 is a selective A2B Adenosine Receptor antagonist. PSB-1115 inhibits the 2,4,6-trinitrobenzenesulfonic acid (TNBS) -induced contraction inhibition of acetylcholine (ACh) [1].

• UNSPSC:

  12352005

• Target:

  Adenosine Receptor

• Type:

  Reference compound

• Related Pathways:

  GPCR/G Protein

• Applications:

  Neuroscience-Neuromodulation

• Field of Research:

  Others

• Assay Protocol:

  https://www.medchemexpress.com/psb-1115.html

• Purity:

  99.0

• Solubility:

  DMSO : 100 mg/mL (ultrasonic) |H2O : 10 mg/mL (ultrasonic; warming; heat to 60°C)

• Smiles:

  O=S (C1=CC=C (C2=NC3=C (NC (N (CCC) C3=O) =O) N2) C=C1) (O) =O

• Molecular Formula:

  C14H14N4O5S

• Molecular Weight:

  350.35

• References & Citations:

  [1]Michael S, et al. Adenosine A (2A) agonist and A (2B) antagonist mediate an inhibition of inflammation-induced contractile disturbance of a rat gastrointestinal preparation. Purinergic Signal. 2010 Mar;6 (1) :117-24.

• Shipping Conditions:

  Blue Ice

• Storage Conditions:

  -20°C (Powder, protect from light)

• Scientific Category:

  Reference compound1

• Clinical Information:

  No Development Reported

• Isoform:

  Adenosine A2B receptor (A2BR)

• CAS Number:

  152529-79-8