PSB-1115

• Description :

  PSB-1115 is a selective A2B Adenosine Receptor antagonist. PSB-1115 inhibits the 2,4,6-trinitrobenzenesulfonic acid (TNBS) -induced contraction inhibition of acetylcholine (ACh) [1].

• UNSPSC :

  12352005

• Target :

  Adenosine Receptor

• Type :

  Reference compound

• Related Pathways :

  GPCR/G Protein

• Applications :

  Neuroscience-Neuromodulation

• Field of Research :

  Others

• Assay Protocol :

  https://www.medchemexpress.com/psb-1115.html

• Purity :

  99.0

• Solubility :

  DMSO : 100 mg/mL (ultrasonic) |H2O : 10 mg/mL (ultrasonic; warming; heat to 60°C)

• Smiles :

  O=S(C1=CC=C(C2=NC3=C(NC(N(CCC)C3=O)=O)N2)C=C1)(O)=O

• Molecular Formula :

  C14H14N4O5S

• Molecular Weight :

  350.35

• References & Citations :

  [1]Michael S, et al. Adenosine A (2A) agonist and A (2B) antagonist mediate an inhibition of inflammation-induced contractile disturbance of a rat gastrointestinal preparation. Purinergic Signal. 2010 Mar;6 (1) :117-24.

• Shipping Conditions :

  Blue Ice

• Storage Conditions :

  -20°C (Powder, protect from light)

• Scientific Category :

  Reference compound1

• Clinical Information :

  No Development Reported

• Isoform :

  Adenosine A2B receptor (A2BR)

• CAS Number :

  [152529-79-8]