WDR5 probe 1

• Description:

  Multi-target kinase-IN-8 is an efficient and highly selective WDR5 chemical probe. Multi-target kinase-IN-8 is a pharmaceutical intermediate. Multi-target kinase-IN-8 can be used for cancer research[1].

• UNSPSC:

  12352005

• Target:

  Drug Intermediate; WDR5

• Related Pathways:

  Epigenetics; Others

• Field of Research:

  Cancer

• Smiles:

  C#CC[C@@H](C(N1CCC2=C(C1)C=CS2)=O)NC(C3=CC(CN4C=CN=C4)=CC(C5=CN(N=C5C(F)(F)F)CC)=C3)=O

• Molecular Formula:

  C29H27F3N6O2S

• Molecular Weight:

  580.62

• References & Citations:

  [1]Hoffmann L, et al. Discovery of an exquisitely selective WDR5 chemical probe accelerated by a high-quality DEL–ML Hit[J]. RSC chemical biology, 2025, 6 (10) : 1585-1594.

• Shipping Conditions:

  Room temperature

• Scientific Category:

  Reference compound1

• Clinical Information:

  No Development Reported