WDR5-MYC-IN-1
CAT:
804-HY-163774
Size:
Inquire
Price:
Ask
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No

WDR5-MYC-IN-1
- UNSPSC Description: WDR5-MYC-IN-1 (compound 4o) is a potent WDR5-MYC interaction inhibitor with a Ki value of 1.0 µM. WDR5-MYC-IN-1 shows antiproliferative activity[1].
- Target Antigen: Histone Methyltransferase
- Type: Reference compound
- Related Pathways: Epigenetics
- Field of Research: Cancer
- Assay Protocol: https://www.medchemexpress.com/wdr5-myc-in-1.html
- Smiles: O=C(NC)C1=CC=C(C2=C(SC#N)SC(N)=N2)C=C1
- Molecular Weight: 290.36
- References & Citations: [1]Wang H, et al. Identification of 5-Thiocyanatothiazol-2-amines Disrupting WDR5-MYC Protein-Protein Interactions. ACS Med Chem Lett. 2024 Jul 1;15(7):1143-1150.
- Shipping Conditions: Room temperature
- Clinical Information: No Development Reported