RJG-2051

CAT: 0804-HY-176084Size: 1 EachDry Ice: NoHazardous: No
CAT#:0804-HY-176084Size:1 Each
Selected
PRICE
AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Product image 1
1 / 1
Description
RJG-2051 is a selective covalent aldo-keto reductase family 1 member C3 (AKR1C3) inhibitor with an IC50 value of 13 nM. RJG-2051 interferes with the metabolic process of substrates such as androgens, estrogens, and prostaglandins by AKR1C3. RJG-2051 is promising for research of cancers[1].
CAS Number
[2851993-77-4]
UNSPSC
12352005
Target
Aldose Reductase
Related Pathways
Metabolic Enzyme/Protease
Field of Research
Cancer
Smiles
COC1=CC=CC=C1N2CCN(CC2)C(C3=CC=C(C=C3)S(=O)(N4C=NC(C5CCCCC5)=N4)=O)=O
Molecular Formula
C26H31N5O4S
Molecular Weight
509.62
References & Citations
[1]Grams RJ, et al. Discovery and Optimization of a Covalent AKR1C3 Inhibitor. J Med Chem. 2025 Apr 25.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported

Related Products

CatalogName
HY-174144RJG-2036
HY-149862-01ARD-2051
HY-133533O-2050
HY-161617LASSBio-2052
HY-19303CRA-2059
HY-D0118A-205
HY-19303B-01CRA-2059 (TFA)
HY-19303ACRA-2059 (hydrochloride)
HY-110020Rel-O-2050
HY-110136-01PMX 205

Alternative Products

CatalogName
C04934RJG-2051
MF-0118158-01RJG-2036
MBS5820583ARD-2051
NBP2-79779-100ugMouse Monoclonal TLE1 Antibody (TLE1/2051)
NBP2-79913BMouse Monoclonal TLE1 Antibody (TLE1/2051) [Biotin]
NBP2-79913PCPMouse Monoclonal TLE1 Antibody (TLE1/2051) [PerCP]
NBP2-79913PEMouse Monoclonal TLE1 Antibody (TLE1/2051) [PE]
NBP2-79913HMouse Monoclonal TLE1 Antibody (TLE1/2051) [HRP]
NBP2-79913FMouse Monoclonal TLE1 Antibody (TLE1/2051) [FITC]
NBP2-79913APCMouse Monoclonal TLE1 Antibody (TLE1/2051) [Allophycocyanin]

Popular Products