NTRC-739

CAT: 0804-HY-12217Size: 1 EachDry Ice: NoHazardous: No
CAT#:0804-HY-12217Size:1 Each
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Description
NTRC-739 is a selective nonpeptide partial neurotensin receptor type 2 (NTS2) agonist with an EC50 of 12 nM and a Ki of 153 nM. NTRC-739 is 161-fold selective for NTS2 versus NTS1. NTRC-739 can be used for the study of chronic pain research[1].
CAS Number
[1612188-96-1]
UNSPSC
12352005
Target
Neurotensin Receptor
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Smiles
O=C(C1(NC(C2=NN(C3=CC=C(F)C=C3)C(C4=CC=CC=C4OC)=C2)=O)CCCCC1)O
Molecular Formula
C24H24FN3O4
Molecular Weight
437.46
References & Citations
[1]Thomas JB, et al. Identification of 1- ({[1- (4-fluorophenyl) -5- (2-methoxyphenyl) -1H-pyrazol-3-yl]carbonyl}amino) cyclohexane carboxylic acid as a selective nonpeptide neurotensin receptor type 2 compound. J Med Chem. 2014 Jun 26;57 (12) :5318-32.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
NTR2

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