CELT-133

CAT: 0931-T83956Size: 10 µgDry Ice: NoHazardous: No
CAT#:0931-T83956Size:10 µg
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Target
Others
Related Pathways
Others
Bioactivity
CELT-133 is a selective fluorescent antagonist for the h?1A adrenergic receptor, demonstrating complete selectivity towards ?1A over ?2A receptors, with a Ki of 5 nM and 15% displacement at 1 ?M in radioligand binding assays, respectively. It displays equivalent affinity across all ?1 adrenergic receptor subtypes. Notably, CELT-133 features excitation and emission maxima (?) at 560 and 571 nm, respectively, making it suitable for use as an acceptor dye in time-resolved Förster resonance energy transfer (TR-FRET) assays when paired with the CoraFluor 1 TR-FRET donor.
Molecular Weight
1318.43
Shipping Conditions
Cool pack
Storage Temperature
-20°C

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