Products for Research Use Only

MSG606 TFA

CAT: 0931-T76003-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0931-T76003-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Target
Melanocortin Receptor
Related Pathways
GPCR/G Protein, Neuroscience
Bioactivity
MSG606 TFA, a potent antagonist of the human MC1 receptor (IC50 = 17 nM), functions as a partial agonist at the human MC3 and MC5 receptors (EC50 values of 59 and 1300 nM, respectively) . It demonstrates binding affinity for A375 melanoma cells in vitro and selectively reverses induced hyperalgesia in female mice without affecting male mice.
Molecular Formula
C63H83F3N20O15S
Molecular Weight
1461.53
Shipping Conditions
Ice Packs
Storage Temperature
-20°C