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Relamorelin TFA

CAT: 0931-T75262-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0931-T75262-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
2863659-22-5
Target
GHSR
Related Pathways
GPCR/G Protein
Bioactivity
Relamorelin (RM-131) TFA, a pentapeptide ghrelin analog, is a potent and selective agonist for the ghrelin/growth hormone secretagogue receptor (GHSR), exhibiting a K_i of 0.42 nM for the GHS-1a receptor. This compound can cross the blood-brain barrier and effectively increases growth hormone levels while promoting faster gastric emptying, showing significant research potential for conditions such as cachexia, gastroparesis, and disorders related to gastric/intestinal motility [1] [2] [3] [4] [5].
Smiles
C(C(O)=O)(F)(F)F.C([C@@H](NC([C@@H](CC=1C=2C(SC1)=CC=CC2)NC(=O)C3CCNCC3)=O)C(N[C@H](C(NC4(C(N)=O)CCNCC4)=O)CC5=CC=CC=C5)=O)C=6C=7C(NC6)=CC=CC7
Molecular Formula
C45H51F3N8O7S
Molecular Weight
905
Shipping Conditions
Ice Packs
Storage Temperature
-20°C