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Relamorelin acetate

CAT: 0931-T39236Size: 25 mgDry Ice: NoHazardous: No
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CAT#:0931-T39236Size:25 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
1809080-14-5
Target
GHSR
Related Pathways
GPCR/G Protein
Bioactivity
Relamorelin (RM-131) acetate is a pentapeptide ghrelin analog that acts as a selective agonist for the ghrelin/growth hormone secretagogue receptor (GHSR) . It exhibits a high affinity for the GHS-1a receptor, with a Ki value of 0.42 nM. Notably, Relamorelin acetate can cross the blood-brain barrier and target the central nervous system. This compound effectively increases growth hormone levels and promotes faster gastric emptying. Due to these properties, Relamorelin acetate holds promise for its potential applications in research related to cachexia, gastroparesis, and gastric/intestinal dysmobility disorders [4] [5].
Smiles
CC(O)=O.NC(=O)C1(CCNCC1)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](Cc1csc2ccccc12)NC(=O)C1CCNCC1
Molecular Formula
C45H54N8O7S
Molecular Weight
851.04
Shipping Conditions
Ice Packs
Storage Temperature
-20°C