Relamorelin

• Target :

  GHSR

• Related Pathways :

  GPCR/G Protein

• Purity :

  >99.99%

• Bioactivity :

  Relamorelin (BIM28131, RM131) is a selective and potent ghrelin/growth hormone secretagogue receptor (GHSR) agonist with high affinity for GHS-1a receptor (Ki value is 0.42 ± 0.063 nM) . Relamorelin (BIM28131, RM131) is also a centrally permeable pentapeptide analog that can increase growth hormone levels and accelerate gastric emptying, and has the potential to study cachexia.

• Smiles :

  C([C@@H](NC([C@@H](CC=1C=2C(SC1)=CC=CC2)NC(=O)C3CCNCC3)=O)C(N[C@H](C(NC4(C(N)=O)CCNCC4)=O)CC5=CC=CC=C5)=O)C=6C=7C(NC6)=CC=CC7

• Molecular Formula :

  C43H50N8O5S

• Molecular Weight :

  790.97

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  661472-41-9