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DPP-4/GPR119 modulator 1

CAT: 0931-T74528-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0931-T74528-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
2411099-68-6
Target
Potassium Channel, Proteasome, GPCR, Others
Related Pathways
Others, Ubiquitination, GPCR/G Protein, Endocrinology/Hormones, Proteases/Proteasome, Membrane transporter/Ion channel
Bioactivity
DPP-4/GPR119 modulator 1 (Compound 22) is an orally active compound that acts as both a dipeptidyl peptidase IV (DPP-IV) inhibitor and GPR119 agonist, demonstrating a glucose-lowering effect in blood and moderate inhibition of the hERG channel with an IC50 value of 4.9 μM. This compound is applicable in diabetes research [1].
Smiles
Cl.CC#CCn1c(nc2n(C)c(=O)n(CCCN3CCN(CC3)c3nc(no3)-c3ccccc3)c(=O)c12)N1CCC[C@@H](N)C1
Molecular Formula
C30H39ClN10O3
Molecular Weight
623.15
Shipping Conditions
Ice Packs
Storage Temperature
-20°C