A2AAR antagonist 4

• Target:

  Adenosine Receptor

• Related Pathways:

  Neuroscience|||GPCR/G Protein

• Bioactivity:

  A2AAR antagonist 4 is an orally active antagonist of the A2A adenosine receptor (A2AAR) with a Ki value of 0.36 nM and a KB value of 1 nM in humans. At a concentration of 10 ?M, it fully inhibits both human A2AAR and human A2bAR. A2AAR antagonist 4 is applicable in cancer research, such as studies involving MC38 tumors.

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C