A2AAR antagonist 3

• Target:

  Adenosine Receptor

• Related Pathways:

  GPCR/G Protein|||Neuroscience

• Bioactivity:

  A2AAR antagonist 3 is a potent and selective A2A adenosine receptor (A2AAR) antagonist with an IC50 value of 1.57 nM. It exhibits a high binding affinity specifically for A2AAR. In vitro studies demonstrate its good stability in rat liver microsomes, and it possesses acceptable pharmacokinetic properties in vivo. A2AAR antagonist 3 is applicable for cancer research.

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C