Products for Research Use Only

PPARγ agonist 19

CAT: 0931-T211307-01Size: 10 mgDry Ice: NoHazardous: No
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CAT#:0931-T211307-01Size:10 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Target
PPAR, COX
Related Pathways
Neuroscience, DNA Damage/DNA Repair, Immunology/Inflammation, Metabolism
Bioactivity
PPARγ agonist19 (Compound 5e) is a PPARγ agonist with an IC50 of 11.27 μM for COX-1 and 0.05 μM for COX-2. It enhances glucose uptake in rat hemidiaphragm assays more effectively than pioglitazone. Additionally, PPARγ agonist19 reduces hyperglycemia and insulin resistance in type 2 diabetic rat models and protects against renal and lipid damage caused by metabolic dysfunction.
Shipping Conditions
Ice Packs
Storage Temperature
-20°C