P-gb-IN-1

• Description:

  P-gb-IN-1 is a potent P-glycoprotein (P-gp) inhibitor that exhibits reverse activity by inhibiting P-gp outflow. P-gb-IN-1 has been shown to inhibit P-gp by hydrogen bonding with residues Asn 721 and Met 986. P-gb-IN-1 showed low toxicity in MCF-7/ADR cells.

• Stability:

  ≥ 2 years

• Purity:

  >98% (HPLC)

• Weight:

  512.55

• Molecular Formula:

  C30H28N2O6

• Notes:

  Research use only, not for human use.

• Receptor:

  P-gp

• CAS Number:

  2632874-49-6