LU-002i (TFA)

CAT: 0804-HY-157034ASize: 1 EachDry Ice: NoHazardous: No
CAT#:0804-HY-157034ASize:1 Each
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
LU-002i TFA is a subunit-selective human proteasome β2c and β2i inhibitor with an IC50 value of 220 nM for β2i[1].
UNSPSC
12352005
Target
Proteasome
Type
Reference compound
Related Pathways
Metabolic Enzyme/Protease
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/lu-002i-tfa.html
Smiles
O=C([C@]1(CO1)C)[C@@H](NC([C@@H](NC([C@H](C)NC(CN2CCOCC2)=O)=O)CC3=CC=C(C=C3)OC)=O)CC4C5([H])C(CCCC5)([H])CCC4.OC(C(F)(F)F)=O
Molecular Formula
C37H53F3N4O9
Molecular Weight
754.83
References & Citations
[1]Xin BT, et al. Structure-Based Design of Inhibitors Selective for Human Proteasome β2c or β2i Subunits. J Med Chem. 2019 Feb 14;62 (3) :1626-1642.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported

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