YK-2168
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No


YK-2168
UNSPSC Description:
YK-2168 is a differentiated selective inhibitor of CDK9[1].Target Antigen:
CDKType:
Reference compoundRelated Pathways:
Cell Cycle/DNA DamageField of Research:
CancerAssay Protocol:
https://www.medchemexpress.com/yk-2168.htmlSmiles:
ClC1=CN=C(NC(C2CCNCC2)=C3)C3=C1C4=CN(C)N=C4Molecular Weight:
315.80References & Citations:
[1]Yingchun Liu, et al. Discovery and preclinical profile of YK-2168, a differentiated selective CDK9 inhibitor in clinical development. Bioorg Med Chem Lett. 2024 Nov 1:112:129941.Yingchun Liu, et al. Discovery and preclinical profile of YK-2168, a differentiated selective CDK9 inhibitor in clinical development. Bioorg Med Chem Lett. 2024 Nov 1:112:129941.Shipping Conditions:
Room temperatureClinical Information:
No Development ReportedCAS Number:
2571068-74-9
