Products for Research Use Only

EGFR-IN-43

CAT: 0013-GTR19221222-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0013-GTR19221222-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
EGFR-IN-43 (Compound 17c) is a potent dual-action inhibitor, covalently linking gefitinib with tamoxifen/endoxifen to simultaneously target EGFR and the estrogen receptor. It exhibits single-digit nanomolar EGFR inhibition and retains ER antagonism, demonstrating promising anti-cancer activity in cellular studies for researching combination therapies in resistant cancers.
Field of Research
Cardiovascular Research, Cell Biology, Signal Transduction
Molecular Formula
C50H55ClFN5O5
Molecular Weight
860.45
Storage Conditions
-20°C
Notes
For research use only.