BAY-299

CAT: 0804-HY-107424-01Size: 5 mgDry Ice: NoHazardous: No
CAT#:0804-HY-107424-01Size:5 mg
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
BAY-299, a chemical probe, is a very potent, dual inhibitor with IC50s of 67 nM for BRPF2 bromodomains (BD), 8 nM for TAF1 BD2, and 106 nM for TAF1L BD2.
CAS Number
[2080306-23-4]
UNSPSC
12352005
Hazard Statement
H302, H315, H319, H335
Target
Epigenetic Reader Domain
Type
Reference compound
Related Pathways
Epigenetics
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/BAY-299.html
Purity
99.40
Solubility
DMSO : 25 mg/mL (ultrasonic; warming)
Smiles
O=C(N1C2=C(C)C=C(N(C)C3=O)C(N3C)=C2)C4=CC=C(CCCO)C5=C4C(C1=O)=CC=C5
Molecular Formula
C25H23N3O4
Molecular Weight
429.47
Precautions
H302, H315, H319, H335
References & Citations
[1]Bouché L, et al. Benzoisoquinolinediones as Potent and Selective Inhibitors of BRPF2 and TAF1/TAF1L Bromodomains. J Med Chem. 2017 May 11;60 (9) :4002-4022.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
BRPF1; BRPF2; BRPF3

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Alternative Products

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406998BAY-299
MBS3603241-01BAY 299
A20239-5BAY-299 5mg
A20239-10BAY-299 10mg
A20239-50BAY-299 50mg
A20239-25BAY-299 25mg
A20239-100BAY-299 100mg
5970/25BAY 299 50 mg
5970/5BAY 299 10 mg
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