BAY-299

• Description:

  BAY-299 is a potent and selective inhibitor of BRD1 and the second bromodomain of TAF1 (Transcription initiation factor TFIID subunits. BAY-299 has IC50values of 6-67 and 8-13 nM for BRD1 and TAF1 inhibitor, respectively. BAY-299 shows selectivity over other bromodomains (>30-fold over other members of the BRPF family; BRD9 and ATAD2; >300-fold over BRD4) .

• Format:

  Solid

• Molecular Formula:

  C25H23N3O4

• Shipping Conditions:

  Room Temperature

• Storage Conditions:

  At least 6 months at -20°C.

• Calculated Molecular Weight:

  429.5 Da

• CAS Number:

  2080306-23-4