DS-3801b

• UNSPSC Description:

  DS-3801b is a potent and non-macrolide agonist of GPR38. DS-3801b is expected to be novel gastrointestinal prokinetic agents for the research of functional gastrointestinal disorders such as gastroparesis and chronic constipation[1].

• Target Antigen:

  Motilin Receptor

• Type:

  Reference compound

• Related Pathways:

  GPCR/G Protein

• Applications:

  Metabolism-protein/nucleotide metabolism

• Field of Research:

  Metabolic Disease

• Assay Protocol:

  https://www.medchemexpress.com/ds-3801b.html

• Solubility:

  DMSO : 100 mg/mL (ultrasonic)

• Smiles:

  O=C([C@H]1CC[C@H](OC2=CC=CC(CO)=C2)CC1)N(C)C3=CC=C(CN4C[C@H](C)NCC4)C(C)=C3

• Molecular Weight:

  465.63

• References & Citations:

  [1]Toda N, et al. Discovery of DS-3801b, a non-macrolide GPR38 agonist with N-methylanilide structure. Bioorg Med Chem Lett. 2022;59:128554.

• Shipping Conditions:

  Room Temperature

• Clinical Information:

  No Development Reported

• CAS Number:

  1369412-66-7