MRS2496

• Description :

  MRS2496 is a selective P2Y1 receptor antagonist with an IC50 value of 1.5 μM, exhibiting antiplatelet aggregation activity. MRS2496 can be used in the research of antiplatelet aggregation and blood-related diseases[1].

• CAS Number :

  [491611-67-7]

• UNSPSC :

  12352005

• Target :

  P2Y Receptor

• Type :

  Reference compound

• Related Pathways :

  GPCR/G Protein

• Field of Research :

  Cardiovascular Disease

• Assay Protocol :

  https://www.medchemexpress.com/mrs2496.html

• Smiles :

  O=P(O)(O)CC(CP(O)(O)=O)CN1C=NC2=C(N=C(N=C12)Cl)NC

• Molecular Formula :

  C10H16ClN5O6P2

• Molecular Weight :

  399.66

• References & Citations :

  [1]Cattaneo M, et al. Antiaggregatory activity in human platelets of potent antagonists of the P2Y 1 receptor. Biochem Pharmacol. 2004 Nov 15;68 (10) :1995-2002. doi: 10.1016/j.bcp.2004.06.026.

• Shipping Conditions :

  Room temperature

• Scientific Category :

  Reference compound1

• Clinical Information :

  No Development Reported

• Isoform :

  P2Y1 Receptor