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CCZ01048 (TFA)

CAT: 0804-HY-P2336A-01Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0804-HY-P2336A-01Size:1 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
CCZ01048 TFA, a α-MSH analogue, exhibits high binding affinity to melanocortin 1 receptor (MC1R) with a Ki of 0.31 nM. CCZ01048 TFA shows rapid internalization into B16F10 melanoma cells and high in vivo stability. CCZ01048 TFA is a promising candidate for PET imaging of malignant melanoma[1].
UNSPSC
12352209
Target
Melanocortin Receptor
Type
Peptides
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/ccz01048-tfa.html
Purity
98.54
Solubility
DMSO : ≥ 100 mg/mL
Smiles
O=C(N[C@H](C(N[C@H](CC1=CC=CC=C1)C(N[C@H](C(N[C@@H](CC2=CNC3=C2C=CC=C3)C(N[C@@H](CCCCNC4=O)C(N)=O)=O)=O)CCCNC(N)=N)=O)=O)CC5=CN=CN5)[C@H](C4)NC([C@H](CCCC)NC(CN6CCC(NC(CN7CCN(CC(O)=O)CCN(CC(O)=O)CCN(CC(O)=O)CC7)=O)CC6)=O)=O.OC(C(F)(F)F)=O
Molecular Formula
C73H106F3N21O18
Molecular Weight
1622.75
References & Citations
[1]Zhang C, et al. Preclinical Melanoma Imaging with 68Ga-Labeled α-Melanocyte-Stimulating Hormone Derivatives Using PET. Theranostics. 2017;7 (4) :805-813. Published 2017 Feb 8.
Shipping Conditions
Blue Ice
Storage Conditions
-80°C, 2 years; -20°C, 1 year (Powder, sealed storage, away from moisture)
Scientific Category
Peptides
Clinical Information
No Development Reported
Isoform
MC1R

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