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AG-041R

CAT: 0804-HY-125314-01Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0804-HY-125314-01Size:1 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
AG-041R is a potent and selective CCK2 Receptor/Gastrin antagonist. AG-041R inhibits gastrin-evoked secretion of pancreastatin with an IC50 of 2.2 nM. AG-041R inhibits cell growth of Mastomys ECL carcinoid tumor cells[1][2].
CAS Number
159883-95-1
UNSPSC
12352005
Target
Cholecystokinin Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Cancer; Endocrinology
Assay Protocol
https://www.medchemexpress.com/ag-041r.html
Solubility
10 mM in DMSO
Smiles
CC(C=C1)=CC=C1NC(C[C@]2(C3=CC=CC=C3N(C2=O)CC(OCC)OCC)NC(NC4=CC=C(C=C4)C)=O)=O
Molecular Formula
C31H36N4O5
Molecular Weight
544.64
References & Citations
[1]Ding XQ, et al. Evaluation of three novel cholecystokinin-B/gastrin receptor antagonists: a study of their effects on rat stomach enterochromaffin-like cell activity. Pharmacol Toxicol. 1997 Nov;81 (5) :232-7.|[2]Lindström, E., et al. Pharmacological analysis of CCK2 receptor antagonists using isolated rat stomach ECL cells. Br. J. Pharmacol. 127 (2), 530-536 (1999) .
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported

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