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GRK2i (TFA)

CAT: 0804-HY-P1396A-01Size: 5 mgDry Ice: NoHazardous: No
CAT#:0804-HY-P1396A-01Size:5 mg
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
GRK2i TFA is a GRK2 inhibitory polypeptide that specifically inhibits Gβγ activation of GRK2. GRK2i TFA corresponds to the Gβγ-binding domain and acts as a cellular Gβγ antagonist[1].
UNSPSC
12352209
Target
G Protein-coupled Receptor Kinase (GRK)
Type
Peptides
Related Pathways
GPCR/G Protein
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/grk2i-tfa.html
Purity
99.89
Solubility
H2O : 100 mg/mL (ultrasonic)
Smiles
O=C([C@@H](N)CC1=CNC2=CC=CC=C12)N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N3[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N4[C@H](C(N[C@H](C(N[C@H](C(O)=O)CO)=O)CCCNC(N)=N)=O)CCC4)=O)CCCCN)=O)CC(N)=O)=O)CCCCN)=O)CCSC)=O)CCCCN)=O)CCC3)=O)C(C)C)=O)CCCNC(N)=N)=O)CCC(N)=O)=O)C(C)C)=O)CC(C)C)=O)CCC(N)=O)=O)CCC(N)=O)=O)C)=O)CCC(O)=O)=O)CCCNC(N)=N)=O)CC5=CC=C(O)C=C5)=O)C)=O)CC(O)=O)=O)CCCNC(N)=N)=O)CC(C)C)=O)CCC(O)=O)=O)CCCCN)=O)CCCCN.OC(C(F)(F)F)=O
Molecular Formula
C152H257F3N50O43S
Molecular Weight
3598.10
References & Citations
[1]Jorge A Sierra-Fonseca, et al. Nerve growth factor induces neurite outgrowth of PC12 cells by promoting Gβγ-microtubule interaction. BMC Neurosci. 2014 Dec 31;15:132.
Shipping Conditions
Blue Ice
Storage Conditions
-80°C, 2 years; -20°C, 1 year (Powder, sealed storage, away from moisture)
Scientific Category
Peptides
Clinical Information
No Development Reported
Isoform
GRK2

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