GRK2i

CAT: 0804-HY-P1396Size: 1 EachDry Ice: NoHazardous: No
CAT#:0804-HY-P1396Size:1 Each
Selected
PRICE
AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Product image 1
1 / 1
Description
GRK2i is a Gβγ-inhibitory peptide that selectively prevents Gβγ-mediated signaling. GRK2i corresponds to the Gβγ-binding domain of GRK2 (G-protein-coupled receptor kinase 2) [1].
CAS Number
[148505-03-7]
UNSPSC
12352209
Target
G Protein-coupled Receptor Kinase (GRK)
Type
Peptides
Related Pathways
GPCR/G Protein
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/grk2i.html
Solubility
10 mM in DMSO
Smiles
O=C(N[C@@H](CCCCN)C(N[C@@H](CCCCN)C(N[C@@H](CCC(O)=O)C(N[C@@H](CC(C)C)C(N[C@@H](CCCNC(N)=N)C(N[C@@H](CC(O)=O)C(N[C@@H](C)C(N[C@@H](CC1=CC=C(C=C1)O)C(N[C@@H](CCCNC(N)=N)C(N[C@@H](CCC(O)=O)C(N[C@@H](C)C(N[C@@H](CCC(N)=O)C(N[C@@H](CCC(N)=O)C(N[C@@H](CC(C)C)C(N[C@@H](C(C)C)C(N[C@@H](CCC(N)=O)C(N[C@@H](CCCNC(N)=N)C(N[C@@H](C(C)C)C(N2[C@@H](CCC2)C(N[C@@H](CCCCN)C(N[C@@H](CCSC)C(N[C@@H](CCCCN)C(N[C@@H](CC(N)=O)C(N[C@@H](CCCCN)C(N3[C@@H](CCC3)C(N[C@@H](CCCNC(N)=N)C(N[C@@H](CO)C(O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)[C@H](CC4=CNC5=CC=CC=C45)N
Molecular Formula
C153H256N50O41S
Molecular Weight
3484.08
References & Citations
[1]Jorge A Sierra-Fonseca, et al. Nerve growth factor induces neurite outgrowth of PC12 cells by promoting Gβγ-microtubule interaction. BMC Neurosci. 2014 Dec 31;15:132.
Shipping Conditions
Room temperature
Scientific Category
Peptides
Clinical Information
No Development Reported
Isoform
GRK2

Related Products

CatalogName
HY-123538-01GRK2 Inhibitor 1
HY-177948GRK2 degrader-1
HY-156863-01GRK2 Inhibitor 2
HY-P84209-01GRK2 Antibody (YA3906, Mouse)
HY-P85534GRK2 Antibody (YA5226, Mouse)
HY-P83204-01GRK2 Antibody (YA2949, Rabbit)
HY-P85193GRK2 Antibody (YA4885, Rabbit)
HY-RS16845Grk2 Mouse Pre-designed siRNA Set A
HY-RS23286Grk2 Rat Pre-designed siRNA Set A
HY-RS05813GRK2 Human Pre-designed siRNA Set A

Alternative Products

CatalogName
MBS5764022GRK2i
T75935-01GRK2i TFA

Popular Products