Products for Research Use Only
RegisterLogin

EP3 antagonist 3

CAT: 0804-HY-147226-01Size: 5 mgDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0804-HY-147226-01Size:5 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
Description
EP3 antagonist 3 (compound 2) is an orally active, potent and selective EP3 antagonist, with a pKi of 8.3. EP3 antagonist 3 shows excellent pharmacokinetic properties. EP3 antagonist 3 can be used for overactive bladder (OAB) research[1].
CAS Number
1227827-88-4
UNSPSC
12352005
Target
Prostaglandin Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Endocrinology; Neurological Disease
Assay Protocol
https://www.medchemexpress.com/ep3-antagonist-3.html
Concentration
10mM
Purity
99.52
Solubility
DMSO : 250 mg/mL (ultrasonic)
Smiles
O=C1OC(C2=CC=C(C3=CC4=C(C=CC=C4)C=C3)NC2=O)(C(C)C)C(N1)=O
Molecular Formula
C21H18N2O4
Molecular Weight
362.38
References & Citations
[1]Jin J, et al. Novel 3-Oxazolidinedione-6-aryl-pyridinones as Potent, Selective, and Orally Active EP3 Receptor Antagonists. ACS Med Chem Lett. 2010 May 14;1 (7) :316-20.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
EP

Related Products

CatalogName
HY-131664EP3 antagonist 2
HY-157496EP3 antagonist 7
HY-157494EP3 antagonist 5
HY-157495EP3 antagonist 6
HY-153256EP3 antagonist 4
HY-P5702EP3
HY-136152MCHR1 antagonist 3
HY-144127-01AR antagonist 3
HY-120652-01A3AR antagonist 3
HY-157303SSTR5 antagonist 3

Alternative Products

CatalogName
TBI2441-250MGPranlukast, Leukotriene CysLT1 antagonist; GPR17 antagonist
TBI2597-50MGMontelukast, Leukotriene CysLT1 antagonist; GPR17 antagonist
cyt-538-01chGH Antagonist
cyt-215-01oGH Antagonist
4031352.0500VIP Antagonist
H-8650.0005PDGF Antagonist
JLB39188-01Vasopressin antagonist
254641Antagonist G
T36127-01TNF-α Antagonist
sc-221406BCCR4 Antagonist

Popular Products